SCHEMBL6960488

SCHEMBL6960488

COc1cc(C)c(C)cc1NC(=S)N1CCN(c2cc(Cl)cc(Cl)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 3/20 0.55
KMT2A Q03164 2/20 0.55
RAB9A P51151 1/20 0.55
DUSP3 P51452 1/20 0.55
PTPN11 Q06124 1/20 0.55
POLB P06746 2/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 4/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAPT P10636 3/20 0.52
CYP3A4 P08684 1/20 0.50
CYP2C19 P33261 1/20 0.50
HPGD P15428 1/20 0.50
MAPK1 P28482 1/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962355 0.89 MAPT (0.50) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6780980 0.89 KDM4E (0.61) KMT2ARAB9APOLBMEN1ALDH1A1
SCHEMBL6955540 0.88 PHGDH (0.49) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6786898 0.88 CYP3A4 (0.55) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6783848 0.87 KMT2A (0.63) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6782920 0.86 KMT2A (0.53) KMT2ARAB9ADUSP3PTPN11POLB
SCHEMBL6780561 0.84 MEN1 (0.73) KMT2APOLBMEN1ALDH1A1SMN1; SMN2
SCHEMBL6782760 0.84 CYP3A4 (0.66) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6652246 0.82 PHGDH (0.55) PHGDHKMT2APOLBMEN1ALDH1A1
SCHEMBL6956652 0.81 KMT2A (0.61) PHGDHKMT2ARAB9ADUSP3PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed