SCHEMBL6955540

SCHEMBL6955540

COc1cc(C)c(C(C)O)cc1NC(=S)N1CCN(c2cc(Cl)cc(Cl)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 3/20 0.49
KMT2A Q03164 2/20 0.48
RAB9A P51151 1/20 0.48
DUSP3 P51452 1/20 0.48
PTPN11 Q06124 1/20 0.48
ALDH1A1 P00352 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 2/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 3/20 0.46
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
GAA P10253 1/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966490 0.90 KMT2A (0.48) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6963684 0.89 MEN1 (0.55) PHGDHKMT2AALDH1A1POLBMEN1
SCHEMBL6960488 0.88 PHGDH (0.55) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6962355 0.82 MAPT (0.50) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6960712 0.79 RBP4 (0.47) KMT2ARAB9AALDH1A1SMN1; SMN2POLB
SCHEMBL6965253 0.78 RBP4 (0.49) KMT2AALDH1A1POLBMAPTMAPK1
SCHEMBL6780980 0.78 KDM4E (0.61) KMT2ARAB9AALDH1A1SMN1; SMN2POLB
SCHEMBL6786898 0.77 CYP3A4 (0.55) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6783848 0.76 KMT2A (0.63) PHGDHKMT2ARAB9ADUSP3PTPN11
SCHEMBL6782920 0.75 KMT2A (0.53) KMT2ARAB9ADUSP3PTPN11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed