Iodide

Iodide

SCHEMBL6962652

I.NC(=Nc1ccc(CCNC(=O)Nc2ccccc2)cc1)c1cccs1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 6/20 0.56
NOS3 P29474 3/20 0.55
NOS2 P35228 2/20 0.55
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA9 Q16790 1/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
FPR2 P25090 1/20 0.49
CNR1 P21554 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038718 0.99 NOS1 (0.57) NOS1NOS3NOS2HDAC1HDAC2
Iodide SCHEMBL4397802 0.88 CNR1 (0.55) NOS1NOS3NOS2HDAC1HDAC2
Iodide SCHEMBL4397806 0.88 CNR1 (0.55) NOS1NOS3NOS2HDAC1HDAC2
SCHEMBL4409778 0.87 CNR1 (0.56) NOS1NOS3NOS2HDAC1HDAC2
SCHEMBL4409780 0.87 CNR1 (0.56) NOS1NOS3NOS2HDAC1HDAC2
SCHEMBL7081205 0.84 NOS1 (0.66) NOS1NOS3NOS2NPC1RAB9A
SCHEMBL6957505 0.84 NPC1 (0.60) NOS1NOS3NOS2NPC1RAB9A
SCHEMBL6969350 0.83 NOS1 (0.63) NOS1NOS3NOS2CA1CA2
SCHEMBL6958481 0.82 NOS1 (0.62) NOS1NOS3NOS2NPC1RAB9A
SCHEMBL6962660 0.82 NOS1 (0.59) NOS1NOS3NOS2HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed