SCHEMBL6962836

SCHEMBL6962836

Cc1csc2c(F)cc(F)cc12

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 1/20 0.34
CYP2A6 P11509 1/20 0.33
KCNA3 P22001 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3483833 0.80 ESR1 (0.34) CYP2A6KCNA3
Hydrochloric Acid SCHEMBL10483651 0.79 CYP2A6 (0.31) CYP2A6
SCHEMBL3483738 0.77 TAAR1 (0.38) CYP2A6
Hydrochloric Acid SCHEMBL10483744 0.74
SCHEMBL10483658 0.73 TSHR (0.40)
SCHEMBL288465 0.71 ACHE (0.39) CYP2A6KCNA3
SCHEMBL31152165 0.71 CYP2A6 (0.39) CYP2A6
SCHEMBL3484364 0.70
SCHEMBL4877866 0.67 CYP2A6 (0.60) CYP2A6
SCHEMBL24898065 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed