SCHEMBL6963407

SCHEMBL6963407

CC(C)c1nc(C2CC2)c(CO[Si](C)(C)C(C)(C)C)c(-c2ccc(F)cc2)c1CO

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GCGR P47871 19/20 0.54
PRKAA2 P54646 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6953314 0.90 GCGR (0.54) GCGRPRKAA2
SCHEMBL2648300 0.88 GCGR (0.70) GCGR
SCHEMBL6961560 0.86 GCGR (0.74) GCGRPRKAA2
SCHEMBL9269790 0.83 GCGR (0.46) GCGRPRKAA2
SCHEMBL6962930 0.81 GCGR (0.74) GCGRPRKAA2
SCHEMBL6961362 0.81 GCGR (0.35) GCGRPRKAA2
SCHEMBL9743369 0.80 GCGR (0.56) GCGR
SCHEMBL8949900 0.80 GCGR (0.62) GCGRPRKAA2
SCHEMBL2662912 0.80 PRKAA2 (0.45) GCGRPRKAA2
SCHEMBL6639179 0.77 GCGR (0.53) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325130-B1 Substituted pyridines BAYER AG (DE) 2003-11-05 EP disclosed
EP-1123924-A1 Substituted pyridines as HMG-COA reductase inhibitors BAYER AG (DE) 2001-08-16 EP disclosed
EP-1123925-A1 Process for preparation of substituted pyridines BAYER AG (DE) 2001-08-16 EP disclosed
CN-1274719-A Process for preparation of substituted pyridine compound BAYER AG (DE) 2000-11-29 CN disclosed
CN-1055684-C Process for preparing substituted pyridine compounds BAYER AG (DE) 2000-08-23 CN disclosed
US-5401746-A FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND HMG-COA REDUCTASE BAYER AKTIENGESELLSCHAFT (DE) 1995-03-28 US disclosed
US-5169857-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1992-12-08 US disclosed
US-5006530-A Certain 7-[2,6-diisopropyl-4-phenyl-5-lower alkoxymethyl-pyrid-3-yl]-3,5-dihydroxy-6-enoates and derivatives useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1991-04-09 US disclosed
CN-1034364-A Substituted pyridines and process for their preparation BAYER AG (DE) 1989-08-02 CN disclosed