SCHEMBL6963665

SCHEMBL6963665

C[C@@H](NCCc1ccc(NC(=N)c2cccs2)cc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 5/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.41
MAPT P10636 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.40
TP53 P04637 2/20 0.40
CYP3A4 P08684 2/20 0.39
LMNA P02545 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27359221 1.00 HTT (0.42) HTTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL9037368 1.00 HTT (0.42) HTTSMN1; SMN2NPC1RAB9AMAPT
Hydrochloric Acid SCHEMBL8597752 0.99 HTT (0.44) HTTSMN1; SMN2NPC1RAB9AMAPT
Hydrochloric Acid SCHEMBL6969614 0.99 HTT (0.44) HTTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL9038599 0.87 NPC1 (0.41) SMN1; SMN2NPC1RAB9AMAPTNFKB1
Bromide SCHEMBL6968763 0.86 NPC1 (0.41) SMN1; SMN2NPC1RAB9AMAPTNFKB1
Hydrochloric Acid SCHEMBL9212801 0.86 NPC1 (0.41) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL6954653 0.82 NPC1 (0.41) HTTSMN1; SMN2NPC1MAPTHPGD
SCHEMBL9037372 0.82 NPC1 (0.51) SMN1; SMN2NPC1RAB9AMAPTHPGD
SCHEMBL6966852 0.80 NPC1 (0.44) SMN1; SMN2NPC1RAB9AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP claimed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed