SCHEMBL6964510

SCHEMBL6964510

O=C(O)c1ccc(CN2C(=O)c3ccccc3C2=O)o1

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.65
POLB P06746 2/20 0.65
KMT2A Q03164 4/20 0.52
TDP1 Q9NUW8 1/20 0.50
HTT P42858 1/20 0.50
MEN1 O00255 2/20 0.49
HPGD P15428 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
CASP3 P42574 1/20 0.49
CA12 O43570 1/20 0.49
CA9 Q16790 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31751926 1.00 ALDH1A1 (0.65) ALDH1A1POLBKMT2ATDP1HTT
SCHEMBL5064689 0.80 ALDH1A1 (0.59) ALDH1A1POLBKMT2ATDP1MEN1
SCHEMBL10743632 0.79 ALDH1A1 (0.55) ALDH1A1POLBKMT2AHTTMEN1
SCHEMBL5460713 0.76 ALDH1A1 (0.57) ALDH1A1POLBKMT2AHTTMEN1
SCHEMBL31753078 0.76 KMT2A (0.74) POLBKMT2AMEN1HPGDHDAC1
SCHEMBL11364469 0.76 ALDH1A1 (0.55) ALDH1A1POLBKMT2AHTTMEN1
SCHEMBL916927 0.76 KMT2A (0.74) POLBKMT2AMEN1HPGDHDAC1
SCHEMBL10179102 0.73 ALDH1A1 (0.49) ALDH1A1POLBKMT2AHTTMEN1
SCHEMBL1680781 0.73 ALDH1A1 (0.46) ALDH1A1POLBKMT2AMEN1HPGD
SCHEMBL6701969 0.72 ALDH1A1 (0.48) ALDH1A1POLBKMT2AHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060178-B1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF ROTAMASE ENZYMES PFIZER (US) 2003-09-03 EP disclosed
US-6610707-B1 Moderate neuronal regeneration and outgrowth and can be used for treating neurological disorders arising from neurodegenerative diseases and nerve damage. PFIZER INC. 2003-08-26 US disclosed
EP-1060178-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF ROTAMASE ENZYMES PFIZER INC. (US) 2000-12-20 EP disclosed
WO-1999045006-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF ROTAMASE ENZYMES PFIZER INC. (US) 1999-09-10 WO disclosed