SCHEMBL6964618

SCHEMBL6964618

CN(C)CCc1c[nH]c2ccc(C3=CCN(C(=O)OC(C)(C)C)CC3)cc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 15/20 0.66
HTR1B P28222 13/20 0.66
GABRP O00591 1/20 0.47
GABRD O14764 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
GABRB2 P47870 1/20 0.47
GABRA4 P48169 1/20 0.47
GABRE P78334 1/20 0.47
GABRA6 Q16445 1/20 0.47
GABRG1 Q8N1C3 1/20 0.47
GABRG3 Q99928 1/20 0.47
GABRQ Q9UN88 1/20 0.47
KMT2A Q03164 1/20 0.46
HTR1A P08908 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29555807 0.90 HTR1D (0.51) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL19839278 0.90 HTR1D (0.51) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL19761221 0.89 GABRP (0.51) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL29555827 0.89 GABRP (0.51) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL19839256 0.85 HTR1D (0.55) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL19838370 0.85 GABRP (0.48) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL19838459 0.85 GABRP (0.48) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL29555714 0.85 GABRP (0.48) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL29555870 0.85 GABRP (0.48) HTR1DHTR1BGABRPGABRDGABRA1
SCHEMBL29555912 0.85 HTR1D (0.55) HTR1DHTR1BGABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed