SCHEMBL696537

SCHEMBL696537

CC(C)(C)C(=O)[C@@H]1C[C@@H](S(=O)(=O)c2ccc(Cl)cc2Cl)CN1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.35
HSD11B1 P28845 1/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
AKR1B1 P15121 1/20 0.34
FLT1 P17948 2/20 0.34
FLT4 P35916 2/20 0.34
KDR P35968 2/20 0.34
HTT P42858 2/20 0.33
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSK P43235 2/20 0.33
CCR2 P41597 1/20 0.33
SLC6A3 Q01959 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
ITGA1 P56199 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2105653 0.87 GRIK1 (0.41) AKR1B1ITGA1GRIK1GRIA2
SCHEMBL2106278 0.78 GRIK1 (0.39) CTSSCTSLCTSBCTSKGAA
SCHEMBL695486 0.75 CTSS (0.63) CTSSCTSLCTSBCTSK
SCHEMBL15170415 0.75 MEN1 (0.38) CTSSHSD11B1HTTCTSLMEN1
SCHEMBL696063 0.75 AKR1B1 (0.40) CTSSHSD11B1AKR1B1CTSLGRIK1
SCHEMBL15173261 0.75 GRIK1 (0.42) CTSSFLT1FLT4KDRCTSL
Hydrochloric Acid SCHEMBL695249 0.74 CTSS (0.62) CTSSCTSLCTSBCTSK
SCHEMBL3716343 0.73 CYP1A2 (0.39) HSD11B1GRIK1GRIA2
SCHEMBL695605 0.73 CTSS (0.37) CTSSHSD11B1AKR1B1CTSLCTSB
SCHEMBL3064422 0.71 CTSS (0.47) CTSSCTSLCTSBCTSKGRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP claimed