SCHEMBL6968434

SCHEMBL6968434

COc1ccc(-c2sc3cc(OC)ccc3c2C(=O)c2ccc(OCc3ccc(F)cc3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 12/20 0.60
ESR2 Q92731 11/20 0.60
TUBB4A P04350 2/20 0.58
TUBB P07437 2/20 0.58
TUBA3C P0DPH7 2/20 0.58
TUBA1B P68363 2/20 0.58
TUBA4A P68366 2/20 0.58
TUBB4B P68371 2/20 0.58
TUBB3 Q13509 2/20 0.58
TUBB2A Q13885 2/20 0.58
TUBB8 Q3ZCM7 2/20 0.58
TUBA3E Q6PEY2 2/20 0.58
TUBA1A Q71U36 2/20 0.58
TUBA1C Q9BQE3 2/20 0.58
TUBB6 Q9BUF5 2/20 0.58
TUBB2B Q9BVA1 2/20 0.58
TUBB1 Q9H4B7 2/20 0.58
CNR1 P21554 1/20 0.57
CNR2 P34972 1/20 0.57
ENPP3 O14638 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970121 0.95 ESR1 (0.66) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL7098723 0.90 CNR1 (0.69) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL6976042 0.89 ESR1 (0.61) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL16346143 0.88 ESR1 (0.57) ESR1ESR2CNR1CNR2ENPP3
SCHEMBL30619809 0.87 ESR1 (0.64) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL26625327 0.87 ESR1 (0.64) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL6981284 0.85 TUBB4A (0.60) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL5026252 0.84 CNR1 (0.78) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL31683596 0.84 TUBB4A (0.60) ESR1ESR2TUBB4ATUBBTUBA3C
SCHEMBL26625282 0.84 TUBB4A (0.60) ESR1ESR2TUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832888-B1 Benzothiophene compounds, compositions, and methods LILLY CO ELI (US) 2003-07-23 EP disclosed
US-5981570-A INHIBITING BONE LOSS OR BONE RESORPTION, PARTICULARLY OSTEOPOROSIS, CARDIOVASCULAR-RELATED PATHOLOGICAL CONDITIONS, INCLUDING HYPERLIPIDEMIA. ELI LILLY AND COMPANY (US) 1999-11-09 US disclosed
EP-0832888-A1 Benzothiophene compounds, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed