SCHEMBL6969188

SCHEMBL6969188

COCCN1CCN(C(=O)OC(C)(C)C)CC1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.49
NR1H2 P55055 2/20 0.42
USP2 O75604 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ESR2 Q92731 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
PARP1 P09874 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
DTYMK P23919 1/20 0.36
TP53 P04637 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12523828 0.92 P2RX7 (0.43) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL28701145 0.86 ADORA1 (0.38) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL4005175 0.86 NR1H2 (0.41) NR1H2USP2SMN1; SMN2ESR2ALDH1A1
SCHEMBL1583253 0.86 P2RX7 (0.46) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL28705739 0.85 MAPK1 (0.38) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL24744821 0.84 NR1H2 (0.40) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL1176507 0.84 NR1H2 (0.40) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL4390630 0.84 NR1H2 (0.41) NR1H2USP2SMN1; SMN2ESR2ALDH1A1
SCHEMBL19034775 0.84 P2RX7 (0.38) P2RX7NR1H2USP2SMN1; SMN2ESR2
SCHEMBL1583540 0.83 CNR2 (0.40) P2RX7NR1H2USP2SMN1; SMN2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882041-B1 PIPERAZINONEPHENYLOXAZOLIDINONE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2003-03-26 EP disclosed
US-6069145-A AGAINST ANTIBIOTIC RESISTANT BACTERIA ZENECA LIMITED (GB) 2000-05-30 US disclosed
EP-0882041-A1 PIPERAZINONEPHENYLOXAZOLIDINONE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS AstraZeneca AB (SE) 1998-12-09 EP disclosed
WO-1997027188-A1 PIPERAZINONEPHENYLOXAZOLIDINONE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS ZENECA LIMITED (GB) 1997-07-31 WO disclosed