SCHEMBL6969945

SCHEMBL6969945

CC(C)c1nc(CCO)n(Cc2ccncc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.34
TDP1 Q9NUW8 1/20 0.32
ENPP2 Q13822 2/20 0.32
GSK3B P49841 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
SOS1 Q07889 1/20 0.31
TLR8 Q9NR97 1/20 0.31
HSP90B1 P14625 1/20 0.31
TRAP1 Q12931 1/20 0.31
PIM1 P11309 1/20 0.30
PIM3 Q86V86 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbamic Acid SCHEMBL5064953 0.94 PIM1 (0.35) KCNH2TDP1ENPP2GSK3BMEN1
SCHEMBL6966489 0.94 TLR8 (0.35) KCNH2TDP1ENPP2GSK3BTLR8
SCHEMBL7086072 0.92 HSP90B1 (0.32) HSP90B1TRAP1
SCHEMBL5852651 0.91 KCNH2 (0.35) KCNH2TDP1MEN1KMT2ASOS1
SCHEMBL6959029 0.91 IDO1 (0.35) KCNH2TDP1GSK3BMEN1KMT2A
SCHEMBL6971862 0.90 HSP90B1 (0.34) GSK3BHSP90B1TRAP1
SCHEMBL7082703 0.89 KCNH2 (0.34) KCNH2TDP1GSK3BHSP90B1TRAP1
SCHEMBL6972780 0.89 MEN1 (0.33) KCNH2ENPP2GSK3BMEN1KMT2A
SCHEMBL7087528 0.89 SRC (0.35) TDP1MEN1KMT2APKM
SCHEMBL6961597 0.88 HSP90B1 (0.32) TDP1TLR8HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed