SCHEMBL6966489

SCHEMBL6966489

CC(C)c1nc(CCCO)n(Cc2ccncc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 7/20 0.35
GSK3B P49841 1/20 0.34
HSP90B1 P14625 1/20 0.33
TRAP1 Q12931 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 1/20 0.33
KCNH2 Q12809 1/20 0.33
TLR7 Q9NYK1 2/20 0.32
ENPP2 Q13822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969945 0.94 KCNH2 (0.34) TLR8GSK3BHSP90B1TRAP1TDP1
SCHEMBL6965157 0.92 TLR8 (0.34) TLR8GSK3BHSP90B1TRAP1TDP1
SCHEMBL6965579 0.91 HSP90B1 (0.35) TLR8GSK3BHSP90B1TRAP1
SCHEMBL7083480 0.91 TLR8 (0.37) TLR8GSK3BTDP1ALDH1A1KCNH2
SCHEMBL6965525 0.90 GSK3B (0.34) GSK3BTDP1ALDH1A1KCNH2TLR7
SCHEMBL5852651 0.89 KCNH2 (0.35) HSP90B1TRAP1TDP1KCNH2
SCHEMBL6969270 0.89 TLR7 (0.35) TLR8GSK3BTDP1ALDH1A1TLR7
SCHEMBL6969774 0.89 ENPP2 (0.35) GSK3BTDP1ALDH1A1TLR7ENPP2
SCHEMBL6974486 0.89 TLR8 (0.35) TLR8HSP90B1TRAP1TDP1ALDH1A1
Carbamic Acid SCHEMBL5064953 0.88 PIM1 (0.35) GSK3BTDP1KCNH2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed