SCHEMBL6971528

SCHEMBL6971528

[CH2]Oc1cc2ccccc2cn1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
CYP2A6 P11509 1/20 0.48
PDPK1 O15530 1/20 0.48
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42
PLAU P00749 1/20 0.40
KDM4E B2RXH2 3/20 0.38
HTR3A P46098 1/20 0.37
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
BTK Q06187 1/20 0.36
NOTUM Q6P988 1/20 0.35
DRD3 P35462 1/20 0.35
KCNH2 Q12809 1/20 0.35
NQO2 P16083 1/20 0.34
GPR3 P46089 1/20 0.34
CHEK1 O14757 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11883542 0.82 CYP1A2 (0.52) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL1536432 0.78 KDM4E (0.57) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL30746959 0.78 KDM4E (0.57) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL28859952 0.78 CYP1A2 (0.44) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL13711922 0.75 CYP1A2 (0.45) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL3372681 0.75 CYP1A2 (0.50) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL161864 0.75 CYP1A2 (0.45) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL28704952 0.75 CYP1A2 (0.45) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL21965360 0.74 GABRP (0.51) CYP1A2CYP2A6PDPK1NPC1RAB9A
SCHEMBL13291032 0.74 CYP1A2 (0.48) CYP1A2CYP2A6PDPK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP claimed
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed