SCHEMBL6971558

SCHEMBL6971558

CCOC(=O)c1ccccc1OC([O])=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.67
HSD17B10 Q99714 4/20 0.57
ALDH1A1 P00352 3/20 0.57
MAPT P10636 3/20 0.50
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
CDC25B P30305 2/20 0.49
MEN1 O00255 1/20 0.49
USP2 O75604 1/20 0.49
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
CYP2C19 P33261 1/20 0.49
MAPK10 P53779 1/20 0.49
KMT2A Q03164 1/20 0.49
PTK2B Q14289 1/20 0.49
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
TBXAS1 P24557 1/20 0.48
LMNA P02545 4/20 0.47
L3MBTL1 Q9Y468 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1283310 0.88 TSHR (0.69) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL5155541 0.87 ALDH1A1 (0.69) TSHRHSD17B10ALDH1A1MEN1CYP3A4
SCHEMBL2112994 0.86 TSHR (0.67) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL30186934 0.86 TSHR (0.67) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL4391361 0.86 TSHR (0.67) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL1872604 0.86 TSHR (0.67) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL23646047 0.85 TSHR (0.61) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL8498851 0.85 TSHR (0.65) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL8587612 0.85 TSHR (0.65) TSHRHSD17B10ALDH1A1MAPTCYP1A2
SCHEMBL14384075 0.85 TSHR (0.65) TSHRHSD17B10ALDH1A1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114841-B1 PROCESS FOR PRODUCING POLYARYLATE TEIJIN LTD (JP) 2003-10-08 EP claimed
US-6417291-B1 CONDENSATION POLYMERIZATION AND ESTERIFICATION OF AROMATIC DIOL AND ESTER-FORMING MONOMER; ENDCAPPING WITH SALICYLIC ACID ESTER DERIVATIVE TEIJIN LIMITED (JP) 2002-07-09 US claimed
US-6410777-B1 HALOGEN-FREE TEIJIN LIMITED (JP) 2002-06-25 US claimed
EP-1114841-A1 PROCESS FOR PRODUCING POLYARYLATE TEIJIN LIMITED (JP) 2001-07-11 EP claimed
EP-0980861-A1 SALICYLIC ESTER DERIVATIVES AND PROCESS FOR PRODUCING THE SAME TEIJIN LIMITED (JP) 2000-02-23 EP claimed
EP-1114841-B1 PROCESS FOR PRODUCING POLYARYLATE TEIJIN LTD (JP) 2003-10-08 EP disclosed
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed
US-6417291-B1 CONDENSATION POLYMERIZATION AND ESTERIFICATION OF AROMATIC DIOL AND ESTER-FORMING MONOMER; ENDCAPPING WITH SALICYLIC ACID ESTER DERIVATIVE TEIJIN LIMITED (JP) 2002-07-09 US disclosed
US-6410777-B1 HALOGEN-FREE TEIJIN LIMITED (JP) 2002-06-25 US disclosed
EP-1114841-A1 PROCESS FOR PRODUCING POLYARYLATE TEIJIN LIMITED (JP) 2001-07-11 EP disclosed
EP-0980861-A1 SALICYLIC ESTER DERIVATIVES AND PROCESS FOR PRODUCING THE SAME TEIJIN LIMITED (JP) 2000-02-23 EP disclosed