SCHEMBL6971559

SCHEMBL6971559

COc1ccc(S(=O)(=O)N2CCC(=O)Nc3ccccc32)cc1OC

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.67
PDE4B Q07343 1/20 0.67
PDE4C Q08493 1/20 0.67
PDE4D Q08499 1/20 0.67
TDP1 Q9NUW8 1/20 0.65
HSD17B10 Q99714 2/20 0.54
LMNA P02545 2/20 0.52
USP2 O75604 1/20 0.52
GLA P06280 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
PKM P14618 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 3/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28702267 0.82 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DTDP1
SCHEMBL29482634 0.82 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DTDP1
SCHEMBL4180004 0.81 PDE4A (0.78) PDE4APDE4BPDE4CPDE4DTDP1
SCHEMBL7356297 0.81 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL6957777 0.81 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DTDP1
SCHEMBL8602658 0.80 PDE4A (0.72) PDE4APDE4BPDE4CPDE4DHSD17B10
SCHEMBL5472876 0.78 ALDH1A1 (0.55) TDP1HSD17B10KMT2AMEN1PKM
SCHEMBL5464500 0.76 ALDH1A1 (0.51) TDP1HSD17B10LMNAKMT2AMEN1
SCHEMBL8325887 0.76 PDE4A (0.86) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL7360537 0.74 PDE4A (0.86) PDE4APDE4BPDE4CPDE4DLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed