SCHEMBL6971692

SCHEMBL6971692

Cc1c(C)c2c(c(C)c1N)CC(C)(CC(=O)O)O2

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
ALOX5 P09917 3/20 0.34
PSEN1 P49768 5/20 0.33
NR1I2 O75469 1/20 0.33
GABRA5 P31644 1/20 0.32
GABRB2 P47870 1/20 0.32
PTPN1 P18031 1/20 0.32
GSTO1 P78417 1/20 0.32
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
PDE4A P27815 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8600719 0.84 PTGS1 (0.51) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8878648 0.80 ALOX5 (0.35) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL6977576 0.80
SCHEMBL8719899 0.79 NR1I2 (0.34) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL6975994 0.78
Hydrochloric Acid SCHEMBL8714516 0.78
SCHEMBL8712759 0.77 ALOX5 (0.33) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8719905 0.76 NR1I2 (0.33) ALOX5NR1I2MEN1KMT2A
SCHEMBL8713459 0.76
SCHEMBL9201658 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed