SCHEMBL697227

SCHEMBL697227

COC(=O)c1ccc(C(=O)N2C[C@H](S(=O)(=O)c3ccccc3C(F)(F)F)C[C@H]2C(=O)N(C#N)C2CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.44
CTSL P07711 4/20 0.42
CTSB P07858 4/20 0.42
CTSK P43235 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL696039 0.90 CTSS (0.45) CTSSCTSLCTSBCTSK
SCHEMBL707038 0.85 CTSS (0.46) CTSSCTSLCTSBCTSK
SCHEMBL696265 0.85 CTSS (0.46) CTSSCTSLCTSBCTSK
SCHEMBL696038 0.84 CTSS (0.58) CTSSCTSLCTSBCTSK
SCHEMBL695871 0.82 CTSS (0.65) CTSSCTSLCTSBCTSK
SCHEMBL694273 0.77 CTSS (0.52) CTSSCTSLCTSB
SCHEMBL696327 0.76 CTSS (0.62) CTSSCTSLCTSBCTSK
SCHEMBL695788 0.75 CTSS (0.59) CTSSCTSLCTSBCTSK
SCHEMBL695427 0.75 CTSS (0.59) CTSSCTSLCTSBCTSK
SCHEMBL695840 0.75 CTSS (0.44) CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP claimed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO claimed
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed