SCHEMBL6972632

SCHEMBL6972632

COc1cc(C(=O)N2CCC(=O)Nc3ccccc32)ccc1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.61
ALDH1A1 P00352 2/20 0.55
CRBN Q96SW2 2/20 0.52
PDE4A P27815 1/20 0.50
PDE4B Q07343 1/20 0.50
PDE4C Q08493 1/20 0.50
PDE4D Q08499 1/20 0.50
LMNA P02545 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ROCK2 O75116 1/20 0.47
BRD2 P25440 1/20 0.46
HTT P42858 1/20 0.46
HSD11B1 P28845 2/20 0.46
TUBB4A P04350 1/20 0.45
TUBB P07437 1/20 0.45
TUBA3C P0DPH7 1/20 0.45
TUBA1B P68363 1/20 0.45
TUBA4A P68366 1/20 0.45
TUBB4B P68371 1/20 0.45
TUBB3 Q13509 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016623 0.86 BRD4 (0.63) BRD4ALDH1A1CRBNPDE4APDE4B
SCHEMBL7021672 0.85 BRD4 (0.59) BRD4ALDH1A1CRBNPDE4APDE4B
SCHEMBL6955057 0.84 BRD4 (0.57) BRD4ALDH1A1CRBNPDE4APDE4B
SCHEMBL6966461 0.81 BRD4 (0.65) BRD4ALDH1A1CRBNLMNANPSR1
SCHEMBL7353031 0.77 PDE4A (0.75) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL6201929 0.77 BRD4 (0.60) BRD4ALDH1A1CRBNLMNANPSR1
SCHEMBL23174997 0.77 BRD4 (0.60) BRD4ALDH1A1CRBNLMNANPSR1
SCHEMBL6958949 0.75 AVPR1A (0.58) BRD4ALDH1A1
SCHEMBL6976978 0.75 PDE4A (0.62) BRD4ALDH1A1PDE4APDE4BPDE4C
SCHEMBL6202811 0.74 BRD4 (0.60) BRD4ALDH1A1CRBNLMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed