SCHEMBL6972931

SCHEMBL6972931

CC(C)c1nc(CO)n(Cc2ccccn2)c1Sc1cccc([N+](=O)[O-])c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.44
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
S1PR3 Q99500 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 4/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
ACHE P22303 1/20 0.36
LMNA P02545 2/20 0.35
PKM P14618 1/20 0.35
KDM4E B2RXH2 3/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961655 0.93 CFTR (0.43) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6967115 0.91 CFTR (0.42) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6969838 0.91 CFTR (0.44) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6969925 0.90 CFTR (0.41) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6966286 0.90 CFTR (0.43) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6973370 0.90 CFTR (0.43) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL8346904 0.89 CFTR (0.41) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6974034 0.89 CFTR (0.41) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL8346908 0.89 CFTR (0.41) CFTRCYP1A2CYP3A4S1PR3L3MBTL1
SCHEMBL6961923 0.89 CYP1A2 (0.44) CFTRCYP1A2CYP3A4S1PR3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed