SCHEMBL6969925

SCHEMBL6969925

CC(C)c1nc(COCCO)n(Cc2ccccn2)c1Sc1cccc([N+](=O)[O-])c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.41
S1PR3 Q99500 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALDH1A1 P00352 5/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
MAPT P10636 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
POLB P06746 2/20 0.34
GAA P10253 1/20 0.34
CTSD P07339 1/20 0.34
ACHE P22303 1/20 0.34
GNRHR P30968 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 2/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975425 0.91 CFTR (0.39) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL6961655 0.90 CFTR (0.43) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL7080059 0.90 CFTR (0.38) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL6972931 0.90 CFTR (0.44) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL6967115 0.89 CFTR (0.42) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL7084592 0.88 CFTR (0.41) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL6974553 0.87 HRH1 (0.34) ALDH1A1KDM4E
SCHEMBL6975011 0.87 CFTR (0.41) CFTRS1PR3CYP1A2CYP3A4ALDH1A1
SCHEMBL7083804 0.87 PDE4A (0.36) ALDH1A1MAPTL3MBTL1POLBLMNA
SCHEMBL6960270 0.87 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed