SCHEMBL6972949

SCHEMBL6972949

CCn1c(COC(N)=O)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 1/20 0.37
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SLC6A9 P48067 3/20 0.35
AKR1B1 P15121 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
TYMS P04818 2/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALOX5 P09917 1/20 0.33
PTPN11 Q06124 2/20 0.32
DHFR P00374 2/20 0.32
TRPM5 Q9NZQ8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974816 0.92 ALOX12 (0.36) ALOX12TP53RXFP1SLC6A9AKR1B1
SCHEMBL7081807 0.92 ALOX12 (0.35) ALOX12TP53RXFP1SLC6A9AKR1B1
SCHEMBL7081639 0.91 ALOX12 (0.38) ALOX12TP53RXFP1SLC6A9AKR1B1
SCHEMBL6975636 0.90 ALOX12 (0.36) ALOX12TP53RXFP1SLC6A9AKR1B1
SCHEMBL6962940 0.90 HSP90B1 (0.31) SMN1; SMN2
SCHEMBL6966621 0.90 TDP1 (0.40) TP53RXFP1SLC6A9
SCHEMBL6974700 0.89 ALOX12 (0.35) ALOX12TP53RXFP1SLC6A9AKR1B1
SCHEMBL7078929 0.89 TP53 (0.37) ALOX12TP53RXFP1SLC6A9AKR1B1
SCHEMBL6974432 0.88 EPHX1 (0.35) SLC6A9SMN1; SMN2DHFR
SCHEMBL6967291 0.88 ALOX12 (0.36) ALOX12TP53RXFP1SLC6A9ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed