SCHEMBL6973083

SCHEMBL6973083

O=[N+]([O-])c1ccc(Cl)c2ccncc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.56
HTT P42858 4/20 0.56
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
LMNA P02545 3/20 0.52
POLB P06746 2/20 0.52
ALDH1A1 P00352 3/20 0.51
TDP1 Q9NUW8 4/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CHUK O15111 1/20 0.47
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HIPK2 Q9H2X6 1/20 0.42
PDE7A Q13946 1/20 0.41
CSNK1A1 P48729 1/20 0.40
CSNK1D P48730 1/20 0.40
CSNK1E P49674 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL11813329 0.98 MAPT (0.55) MAPTHTTMEN1KMT2ALMNA
SCHEMBL619318 0.93 MAPT (0.52) MAPTHTTMEN1KMT2ALMNA
SCHEMBL11817125 0.87 MAPT (0.64) MAPTHTTMEN1KMT2ALMNA
SCHEMBL31162406 0.79 MAPT (0.58) MAPTHTTMEN1KMT2ALMNA
SCHEMBL246756 0.79 MAPT (0.58) MAPTHTTMEN1KMT2ALMNA
SCHEMBL26933026 0.77 MAPT (0.54) MAPTHTTMEN1KMT2ALMNA
SCHEMBL197023 0.77 GAA (0.52) LMNAALDH1A1SMN1; SMN2GAACHUK
SCHEMBL13483429 0.76 MAPT (0.52) MAPTHTTMEN1KMT2ALMNA
SCHEMBL3577339 0.76 MAPT (0.52) MAPTHTTMEN1KMT2ALMNA
SCHEMBL5921938 0.76 CTSB (0.61) MAPTHTTMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113861110-B Polysubstituted sulfonamide compound, preparation method and medical application thereof 中国药科大学 2024-03-01 CN disclosed
CN-113861110-A Polysubstituted sulfonamide compound, preparation method and medical application thereof 中国药科大学 2021-12-31 CN disclosed
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed
US-3930837-A 3-CHLORO-5-ACETAMIDAISOQUINOLINE AS A HERBICIDE ICI AUSTRALIA LIMITED (AU) 1976-01-06 US disclosed