SCHEMBL6973312

SCHEMBL6973312

CC(=O)Oc1nc(C(C)C)c(Sc2ccccc2)n1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
TSHR P16473 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 3/20 0.33
CYP19A1 P11511 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
KLKB1 P03952 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
P2RX3 P56373 1/20 0.33
CYP3A4 P08684 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082609 0.89 IDO1 (0.38) KMT2AALDH1A1TDP1KDM4EPTGDR2
SCHEMBL6975519 0.89 ALDH1A1 (0.41) ALDH1A1TDP1SMN1; SMN2KDM4EPTGDR2
SCHEMBL6963163 0.88 GRIN1 (0.36) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL6973011 0.88 MEN1 (0.34) KMT2AMEN1ALDH1A1CYP19A1TDP1
SCHEMBL6964793 0.87 MEN1 (0.33) KMT2AMEN1ALDH1A1CYP19A1SMN1; SMN2
SCHEMBL6973925 0.85 PDE4A (0.37) KMT2AMEN1CYP2C9CYP2C19ALDH1A1
SCHEMBL6960619 0.85 MEN1 (0.37) KMT2AMEN1TSHRCYP1A2CYP2C9
SCHEMBL7084768 0.84 PTGDR2 (0.36) KMT2AMEN1TSHRCYP1A2CYP2C9
SCHEMBL6975584 0.84 TDP1 (0.34) KMT2AMEN1TSHRCYP1A2CYP2C9
SCHEMBL6975053 0.84 MEN1 (0.41) KMT2AMEN1TSHRCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed