SCHEMBL6973790

SCHEMBL6973790

Cc1cc(C)cc(Sc2nc(CO)n(Cc3ccncc3)c2C(C)C)c1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.33
KCNH2 Q12809 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
S1PR3 Q99500 1/20 0.31
PHGDH O43175 1/20 0.31
TYMS P04818 1/20 0.31
P2RX3 P56373 1/20 0.30
BRD4 O60885 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973951 0.90 MEN1 (0.37) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL6968175 0.89 KCNH2 (0.35) MEN1KMT2AKCNH2S1PR3
SCHEMBL6974051 0.88 S1PR3 (0.33) MEN1KMT2AKCNH2HPGDS1PR3
SCHEMBL6973406 0.86 KDM4E (0.36) MEN1KMT2AKDM4EALDH1A1S1PR3
SCHEMBL8113749 0.84 MEN1 (0.34) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL7082932 0.84 CSNK2A2 (0.38) MEN1KMT2AGAAKCNH2KDM4E
SCHEMBL6974317 0.83 GRIN1 (0.36) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL7083001 0.82 MEN1 (0.34) MEN1KMT2AGAAKCNH2KDM4E
SCHEMBL6973695 0.82 DHODH (0.31)
SCHEMBL6973582 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed