SCHEMBL6974317

SCHEMBL6974317

CC(C)c1c(Sc2cccc(F)c2)nc(CO)n1Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
KMT2A Q03164 2/20 0.33
ATM Q13315 1/20 0.33
S1PR3 Q99500 1/20 0.33
CYP3A4 P08684 4/20 0.32
CYP2D6 P10635 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
P2RX3 P56373 2/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
CYP17A1 P05093 1/20 0.32
DHODH Q02127 1/20 0.32
USP2 O75604 2/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974051 0.91 S1PR3 (0.33) GRIN1GRIN2BKMT2AS1PR3MEN1
SCHEMBL6961097 0.90 GRIN1 (0.36) GRIN1GRIN2BLMNATP53KMT2A
SCHEMBL7082932 0.89 CSNK2A2 (0.38) LMNATP53KMT2ACYP3A4CYP2C9
SCHEMBL7086504 0.88 GRIN1 (0.33) GRIN1GRIN2BLMNATP53KMT2A
SCHEMBL6973406 0.87 KDM4E (0.36) KMT2AS1PR3CYP3A4CYP2D6CYP2C9
SCHEMBL7078281 0.86 ENPP2 (0.36) GRIN1GRIN2BLMNATP53S1PR3
SCHEMBL7081063 0.85 ENPP2 (0.35) GRIN1GRIN2BLMNATP53S1PR3
SCHEMBL6969383 0.85 DHODH (0.41) KMT2AATMDHODHCA2CA4
SCHEMBL8109545 0.84 GRIN1 (0.36) GRIN1GRIN2BLMNATP53KMT2A
SCHEMBL6968076 0.84 PDE4A (0.39) LMNAKMT2AATMMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed