SCHEMBL6976478

SCHEMBL6976478

Cc1cc(=O)c(-c2ccc(Cl)c(Cl)c2)c(-c2ccccc2)o1

nearest known ligand 0.72

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.72
PTGS1 P23219 2/20 0.72
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
EPHX2 P34913 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1377981 0.84 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL6969701 0.83 PTGS2 (0.80) PTGS2PTGS1
SCHEMBL9261161 0.80 PTGS2 (0.60) PTGS2PTGS1HTT
SCHEMBL7612769 0.76 PTGS2 (0.48) PTGS2PTGS1RXRARXRBRXRG
SCHEMBL6977125 0.76 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL6972308 0.75 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL1376982 0.75 PTGS2 (0.84) PTGS2PTGS1
SCHEMBL6967436 0.74 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL6973887 0.73 PTGS2 (0.80) PTGS2PTGS1
SCHEMBL6975145 0.71 PTGS2 (0.74) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518303-B2 Selectively inhibit COX-2 in preference to COX-1 and are useful in the treatment of COX-2 mediated diseases, such as inflammation, pain, fever and asthma with fewer side effects ALMIRALL PRODESFARMA S.A. (ES) 2003-02-11 US disclosed
EP-1115716-B1 2-PHENYLPYRAN-4-ONE DERIVATIVES ALMIRALL PRODESFARMA AG (CH) 2003-01-02 EP disclosed