SCHEMBL6977301

SCHEMBL6977301

COc1ccc2c(c1)c(OCCOc1c(F)cc(F)cc1Br)nn2S(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
AKR1C3 P42330 3/20 0.36
AKR1C2 P52895 3/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 2/20 0.34
CA9 Q16790 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975124 0.95 HTR6 (0.39) HTR6CYP3A4CYP2D6PTGDR2MEN1
SCHEMBL6967992 0.92 HTR6 (0.39) HTR6CYP3A4CYP2D6PTGDR2MEN1
SCHEMBL6971624 0.86 HTR6 (0.41) HTR6CYP3A4CYP2D6PTGDR2MEN1
SCHEMBL6966090 0.86 HTR6 (0.44) HTR6PTGS1PTGS2AKR1C3AKR1C2
SCHEMBL6968667 0.84 HTR6 (0.48) HTR6PTGS1PTGS2AKR1C3AKR1C2
SCHEMBL6970702 0.84 HTR6 (0.47) HTR6PTGS1PTGS2AKR1C3AKR1C2
SCHEMBL6975027 0.81 HTR6 (0.45) HTR6PTGS1PTGS2AKR1C3AKR1C2
SCHEMBL6971751 0.81 CNR2 (0.41) HTR6MEN1KMT2A
SCHEMBL6971241 0.80 AKR1C3 (0.46) HTR6PTGS1PTGS2AKR1C3AKR1C2
SCHEMBL6967417 0.79 HTR6 (0.41) HTR6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077947-B1 NOVEL 1,5 AND 3-O-SUBSTITUTED 1H-INDAZOLES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY, IMMUNO-MODULATING AND NEURO-PROTECTIVE EFFECT, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS DRESDEN ARZNEIMITTEL (DE) 2003-09-03 EP claimed