SCHEMBL697835

SCHEMBL697835

CCOc1ccc(COC(=O)n2ccnc2[C@@H](C)c2cccc(C)c2C)cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.41
TP53 P04637 1/20 0.41
CALM1 P0DP23 2/20 0.41
LMNA P02545 5/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
GAA P10253 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADORA2A P29274 1/20 0.37
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
CSF1R P07333 1/20 0.36
TSHR P16473 1/20 0.35
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698141 0.95 KMT2A (0.38) MAPTTP53CALM1LMNASMN1; SMN2
SCHEMBL698178 0.93 SLC22A12 (0.35) MAPTTP53LMNATDP1POLB
SCHEMBL703828 0.92 MEN1 (0.42) MAPTLMNASMN1; SMN2MEN1KMT2A
SCHEMBL697607 0.90 ALKBH1 (0.36) MAPTLMNASMN1; SMN2TDP1ALDH1A1
SCHEMBL697913 0.88 PDE4B (0.40) TDP1CSF1R
SCHEMBL697860 0.87 FFAR1 (0.35) MAPTLMNAPOLB
SCHEMBL699122 0.86 FFAR1 (0.41) MAPTLMNAPOLBMEN1KMT2A
SCHEMBL708924 0.86 FFAR1 (0.38) TP53LMNASMN1; SMN2TDP1CYP3A4
SCHEMBL3533515 0.86 TP53 (0.40) MAPTTP53LMNASMN1; SMN2TDP1
SCHEMBL696627 0.86 GRIN2B (0.40) MAPTLMNASMN1; SMN2TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423199-A1 Substituted imidazoles and their use as pesticides Pfizer Limited (GB) 2012-02-29 EP disclosed
US-7825149-B2 Substituted imidazoles PFIZER LIMITED (GB) 2010-11-02 US disclosed
US-20090312326-A1 SUBSTITUTED IMIDAZOLES PFIZER LIMITED (GB) 2009-12-17 US disclosed
US-7592362-B2 Substituted imidazoles PFIZER LIMITED (GB) 2009-09-22 US disclosed
US-7547718-B2 Substituted imidazoles PFIZER LIMITED (GB) 2009-06-16 US disclosed
US-7544706-B2 Substituted imidazoles PFIZER LIMITED (GB) 2009-06-09 US disclosed
US-20080125473-A1 SUBSTITUTED IMIDAZOLES PFIZER LIMITED (GB) 2008-05-29 US disclosed
US-20080119536-A1 SUBSTITUTED IMIDAZOLES PFIZER LIMITED (GB) 2008-05-22 US disclosed
US-20070167506-A1 SUBSTITUTED IMIDAZOLES PFIZER INC. (US) 2007-07-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080125473-A1 SUBSTITUTED IMIDAZOLES ABL1, TYR, CYP3A4 MAPT 316/4885TP53 2394/4885CALM1 1072/4885
US-20090312326-A1 SUBSTITUTED IMIDAZOLES ABL1, TYR, CYP3A4 MAPT 316/4885TP53 2394/4885CALM1 1072/4885
US-20070167506-A1 SUBSTITUTED IMIDAZOLES ABL1, TYR, CYP3A4 MAPT 316/4885TP53 2394/4885CALM1 1072/4885
US-20080119536-A1 SUBSTITUTED IMIDAZOLES ABL1, TYR, CYP3A4 MAPT 316/4885TP53 2394/4885CALM1 1072/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.