SCHEMBL6978714

SCHEMBL6978714

O=C1NC(=Cc2ccc3cc(O)ccc3c2)C(=O)S1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.54
DYRK1A Q13627 2/20 0.54
CSNK2A2 P19784 1/20 0.54
CLK1 P49759 1/20 0.54
CSNK2B P67870 1/20 0.54
DYRK2 Q92630 1/20 0.54
DYRK1B Q9Y463 1/20 0.54
AKR1B1 P15121 2/20 0.48
TDP1 Q9NUW8 7/20 0.47
GSK3B P49841 4/20 0.47
RAB9A P51151 2/20 0.47
HPGD P15428 1/20 0.47
KDM4E B2RXH2 3/20 0.44
MAPT P10636 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 2/20 0.44
NSD2 O96028 1/20 0.44
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5673273 0.84 TDP1 (0.66) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL1249053 0.82 GSK3B (0.73) CSNK2A1DYRK1AAKR1B1TDP1GSK3B
SCHEMBL1249051 0.82 GSK3B (0.73) CSNK2A1DYRK1AAKR1B1TDP1GSK3B
SCHEMBL7510151 0.73 CSNK2A2 (0.45) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL6785387 0.73 IGF1R (0.67) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL9254370 0.72 PIM1 (0.71) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL7463867 0.72 PIM1 (0.68) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL4156417 0.72 CSNK2A2 (0.65) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL7519991 0.72 CSNK2A2 (0.65) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B
SCHEMBL9376844 0.71 PTPN1 (0.72) CSNK2A1DYRK1ACSNK2A2CLK1CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1186588-A1 6-HYDROXY-2-NAPHTHYLCARBINOL AND PROCESS FOR THE PREPARATION THEREOF MITSUBISHI CHEMICAL CORPORATION (JP) 2002-03-13 EP claimed
JP-10139768-A None JP disclosed
EP-0801063-B1 Thiazolidinedione derivatives having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them REDDYS LAB LTD DR (IN) 2003-01-15 EP disclosed
EP-1186588-A1 6-HYDROXY-2-NAPHTHYLCARBINOL AND PROCESS FOR THE PREPARATION THEREOF MITSUBISHI CHEMICAL CORPORATION (JP) 2002-03-13 EP disclosed
US-5925656-A CONTAINING A 2,4-DIOXOTRIAZOLIDINE RING DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-07-20 US disclosed
JP-H10139768-A PRODUCTION OF NAPHTHALENE DERIVATIVE MITSUBISHI CHEM CORP 1998-05-26 JP disclosed
EP-0801063-A1 Thiazolidinedione derivatives having antidiabetic, hypolipidaemic antihypertensive properties, process for their preparation and pharmaceutical compositions containing them DR. REDDY'S RESEARCH FOUNDATION (IN) 1997-10-15 EP disclosed