SCHEMBL6979190

SCHEMBL6979190

CN(Cc1ccc(C#N)cc1)C(=O)N1CCCc2cc(NS(=O)(=O)c3ccccc3)ccc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 7/20 0.56
ADRB2 P07550 5/20 0.52
ADRB1 P08588 5/20 0.52
ADRB3 P13945 3/20 0.52
MAPT P10636 2/20 0.48
TP53 P04637 1/20 0.48
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6974865 0.86 NR3C1 (0.56) NR3C1ADRB2ADRB1ADRB3MAPT
SCHEMBL6983044 0.83 NR3C1 (0.58) NR3C1ADRB2ADRB1ADRB3MAPT
SCHEMBL6985317 0.83 NR3C1 (0.58) NR3C1ADRB2ADRB1ADRB3MAPT
SCHEMBL6982976 0.83 NR3C1 (0.54) NR3C1ADRB2ADRB1MAPTTP53
SCHEMBL6981761 0.83 LIMK2 (0.40) NR3C1ADRB2ADRB1ADRB3MAPT
SCHEMBL6981758 0.82 NR3C1 (0.56) NR3C1ADRB2ADRB1ADRB3MAPT
SCHEMBL6985366 0.82 NR3C1 (0.66) NR3C1MAPTTP53ALDH1A1LMNA
SCHEMBL6977969 0.82 NR3C1 (0.56) NR3C1ADRB2ADRB1ADRB3MAPT
SCHEMBL6976880 0.81 NR3C1 (0.55) NR3C1MAPTTP53LMNASMN1; SMN2
SCHEMBL6980538 0.80 NR3C1 (0.56) NR3C1MAPTTP53ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1048667-B1 Process for preparing 8-cyclopentyl-6-ethyl-3-(substituted)-5,8-dihydro-4H-1,2,3A,7,8-pentaaza-as-indacenes and intermediates useful therein PFIZER PROD INC (US) 2003-10-22 EP claimed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed