SCHEMBL6980955

SCHEMBL6980955

N#Cc1ccc(CCC(=O)N2CCCc3cc(NS(=O)(=O)c4cccc5cnccc45)ccc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.43
NR3C1 P04150 6/20 0.43
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
PKLR P30613 1/20 0.43
P2RX7 Q99572 5/20 0.42
F2 P00734 1/20 0.41
FLT3 P36888 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977885 0.91 NR3C1 (0.48) NR3C1BRD4CREBBPSMN1; SMN2
Hydrochloric Acid SCHEMBL6979711 0.88 F2 (0.54) ROCK2NR3C1BRD4CREBBPPKLR
SCHEMBL6977631 0.83 BRD4 (0.56) NR3C1BRD4CREBBPSMN1; SMN2
SCHEMBL6977179 0.83 NR3C1 (0.64) NR3C1BRD4CREBBPSMN1; SMN2
SCHEMBL6982493 0.82 NR3C1 (0.50) NR3C1BRD4CREBBPSMN1; SMN2
SCHEMBL7960284 0.82 NR3C1 (0.47) NR3C1BRD4CREBBPSMN1; SMN2
SCHEMBL6985317 0.81 NR3C1 (0.58) NR3C1SMN1; SMN2
SCHEMBL6982160 0.81 NR3C1 (0.61) NR3C1SMN1; SMN2
SCHEMBL6977969 0.79 NR3C1 (0.56) NR3C1SMN1; SMN2
SCHEMBL6978212 0.79 TRIM24 (0.48) NR3C1BRD4CREBBPSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed