SCHEMBL6981734

SCHEMBL6981734

N#Cc1ccc(Cl)cc1OCCC(NCCO)c1ccno1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.40
NOS2 P35228 7/20 0.40
CYP2D6 P10635 6/20 0.40
SLC6A2 P23975 6/20 0.40
KCNH2 Q12809 2/20 0.38
IDH1 O75874 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
S1PR3 Q99500 2/20 0.35
S1PR1 P21453 2/20 0.35
SLC22A12 Q96S37 1/20 0.34
F11 P03951 2/20 0.34
KLKB1 P03952 2/20 0.34
CYP3A4 P08684 1/20 0.34
P2RX3 P56373 1/20 0.32
P2RX2 Q9UBL9 1/20 0.32
F10 P00742 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7608216 0.82 NOS2 (0.42) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL7604665 0.81 NOS2 (0.39) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL7608154 0.80 CYP2D6 (0.40) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL6503984 0.78 NOS2 (0.49) SLC6A4NOS2CYP2D6SLC6A2KCNH2
Oxalic Acid SCHEMBL6504705 0.74 NOS2 (0.53) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL1306764 0.73 IDH1 (0.53) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL6504708 0.71 NOS2 (0.47) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL6489165 0.70 NOS2 (0.50) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL6492130 0.70 NOS2 (0.49) SLC6A4NOS2CYP2D6SLC6A2KCNH2
SCHEMBL6491319 0.70 NOS2 (0.64) SLC6A4NOS2CYP2D6SLC6A2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003523988-A 2003-08-12 JP claimed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP claimed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO claimed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed