SCHEMBL6981967

SCHEMBL6981967

CNC(=O)c1cc(C(=O)c2ccccc2)ccc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.57
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
L3MBTL1 Q9Y468 2/20 0.47
ATM Q13315 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ABCC9 O60706 1/20 0.45
ABCC8 Q09428 1/20 0.45
KCNJ11 Q14654 1/20 0.45
KCNJ8 Q15842 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CDC25A P30304 1/20 0.44
CDC25B P30305 1/20 0.44
HSD17B10 Q99714 1/20 0.44
DHODH Q02127 1/20 0.43
SRD5A2 P31213 1/20 0.43
SERPINE1 P05121 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31052933 0.87 TDP1 (0.57) GAANPC1RAB9AL3MBTL1ATM
SCHEMBL23263412 0.83 GAA (0.55) GAANPC1RAB9AKDM4EALDH1A1
SCHEMBL8606277 0.82 ATM (0.52) NPC1RAB9AL3MBTL1ATMTDP1
SCHEMBL9766594 0.82 ATM (0.52) NPC1RAB9AL3MBTL1ATMTDP1
SCHEMBL9759904 0.81 BRAF (0.55) GAANPC1L3MBTL1ATMTDP1
SCHEMBL9812344 0.81 MEN1 (0.58) GAANPC1RAB9AL3MBTL1ATM
SCHEMBL11357069 0.77 RAB9A (0.62) NPC1RAB9AL3MBTL1ATMTDP1
SCHEMBL9760868 0.77 MAPK1 (0.59) GAATDP1KDM4EALDH1A1MEN1
SCHEMBL332679 0.76 ATM (0.61) NPC1RAB9AL3MBTL1ATMTDP1
SCHEMBL11504870 0.76 AKR1C3 (0.63) GAAATMTDP1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322599-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-02 EP disclosed
WO-2001096283-A9 HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2002-10-17 WO disclosed
WO-2001096283-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-12-20 WO disclosed