SCHEMBL6982071

SCHEMBL6982071

COc1ccc2nc(-c3nc(N)nc(N)n3)sc2c1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.66
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2C19 P33261 1/20 0.63
ILK Q13418 1/20 0.57
GLA P06280 1/20 0.56
GAA P10253 1/20 0.56
PDK1 Q15118 1/20 0.54
NPC1 O15118 1/20 0.52
SULT1A1 P50225 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8125517 0.89 APP (0.54) APPCYP1A2CYP3A4CYP2C19ILK
SCHEMBL229456 0.81 APP (0.68) APPCYP1A2CYP3A4CYP2C19ILK
SCHEMBL2055237 0.80 APP (0.71) APPCYP1A2CYP3A4CYP2C19ILK
SCHEMBL12974045 0.79 APP (1.00) APPCYP1A2CYP3A4CYP2C19GLA
SCHEMBL1977100 0.79 APP (1.00) APPCYP1A2CYP3A4CYP2C19GLA
SCHEMBL5429982 0.78 APP (0.83) APPGLAGAANPC1SULT1A1
SCHEMBL28801433 0.78 APP (0.64) APPCYP1A2CYP3A4CYP2C19ILK
SCHEMBL29683488 0.78 CYP3A4 (1.00) APPCYP1A2CYP3A4CYP2C19GAA
SCHEMBL22358 0.78 CYP3A4 (1.00) APPCYP1A2CYP3A4CYP2C19GAA
SCHEMBL13806286 0.77 APP (0.63) APPCYP1A2CYP3A4CYP2C19ILK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6150362-A ADMINISTERING 1,3,5-SUBSTITUTED TRIAZINE COMPOUNDS TO THE PATIENT SUFFERING FROM ANGIOGENIC DISEASES ABBVIE INC. 2000-11-21 US claimed
EP-1037886-A1 TRIAZINE ANGIOGENESIS INHIBITORS Abbott Laboratories (US) 2000-09-27 EP claimed
WO-1999031088-A1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LABORATORIES (US) 1999-06-24 WO claimed
EP-1037886-B1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LAB (US) 2003-05-02 EP disclosed
US-6288228-B1 DIAMINOTRIAZINE DERIVATIVES ABBOTT LABORATORIES 2001-09-11 US disclosed
US-6150362-A ADMINISTERING 1,3,5-SUBSTITUTED TRIAZINE COMPOUNDS TO THE PATIENT SUFFERING FROM ANGIOGENIC DISEASES ABBVIE INC. 2000-11-21 US disclosed