SCHEMBL6983713

SCHEMBL6983713

CS(=O)(=O)c1ccc(-n2nc(C(F)F)cc2-c2nc3ccc(F)cc3o2)cc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.48
PTGS1 P23219 10/20 0.44
ABCB11 O95342 1/20 0.42
ALDH1A1 P00352 1/20 0.42
AOC3 Q16853 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977701 0.90 PTGS2 (0.52) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6982590 0.85 PTGS2 (0.63) PTGS2PTGS1
SCHEMBL6982553 0.81 PTGS2 (0.46) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8953911 0.78 PTGS2 (0.73) PTGS2PTGS1ABCB11ALDH1A1AOC3
SCHEMBL9003118 0.78 PTGS2 (0.73) PTGS2PTGS1ABCB11ALDH1A1AOC3
SCHEMBL6972326 0.78 PTGS2 (0.48) PTGS2PTGS1ABCB11ALDH1A1AOC3
SCHEMBL6979695 0.76 PTGS2 (0.48) PTGS2PTGS1ABCB11ALDH1A1AOC3
SCHEMBL6984048 0.75 PTGS2 (0.63) PTGS2PTGS1ABCB11
SCHEMBL6982004 0.75 PTGS2 (0.63) PTGS2PTGS1ABCB11
SCHEMBL9002626 0.72 PTGS2 (0.77) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed