SCHEMBL6984157

SCHEMBL6984157

O=C(O)c1sc2cccnc2c1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 2/20 0.50
LMNA P02545 1/20 0.47
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 5/20 0.41
GPR35 Q9HC97 1/20 0.39
MCL1 Q07820 2/20 0.37
NAPRT Q6XQN6 1/20 0.37
L3MBTL1 Q9Y468 3/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.36
KDM6B O15054 1/20 0.36
KDM6A O15550 1/20 0.36
TET3 O43151 1/20 0.36
KDM4A O75164 1/20 0.36
KDM4B O94953 1/20 0.36
KDM5C P41229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10507045 0.78 LIMK1 (0.55) LIMK1LMNACYP2C9CYP2C19KDM4E
SCHEMBL27404716 0.78 LIMK1 (0.55) LIMK1LMNAKDM4EALDH1A1GPR35
SCHEMBL8507168 0.76 LIMK1 (0.77) LIMK1LMNAKDM4EALDH1A1MCL1
SCHEMBL1098450 0.76 LIMK1 (0.54) LIMK1LMNAKDM4EALDH1A1MCL1
SCHEMBL7508777 0.74 CYP2C9 (0.46) LIMK1LMNACYP2C9CYP2C19KDM4E
SCHEMBL13736548 0.74 MCL1 (0.57) LIMK1LMNACYP2C9CYP2C19KDM4E
SCHEMBL2895816 0.73 LIMK1 (0.50) LIMK1LMNAKDM4EALDH1A1GPR35
SCHEMBL4859707 0.73 LIMK1 (0.50) LIMK1LMNAKDM4EALDH1A1MCL1
SCHEMBL29631384 0.72 LIMK1 (0.49) LIMK1LMNAKDM4EALDH1A1GPR35
SCHEMBL21813696 0.72 LIMK1 (0.56) LIMK1LMNACYP2C9CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed