SCHEMBL6984515

SCHEMBL6984515

C1=C(c2cn(-c3ccccc3)c3ccccc23)CCNC1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 14/20 0.64
HTR1A P08908 3/20 0.56
HTR2C P28335 3/20 0.56
DRD3 P35462 2/20 0.56
HTR7 P34969 2/20 0.56
HTR2A P28223 2/20 0.56
DRD2 P14416 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
ALOX15 P16050 1/20 0.49
HSD17B10 Q99714 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
KHK P50053 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10874677 0.90 HTR6 (0.57) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL16260562 0.90 HTR6 (0.56) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL14406061 0.86 HTR6 (0.56) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL7138867 0.80 HTR6 (0.60) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL27557297 0.80 HTR6 (0.60) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL27336067 0.80 HTR6 (0.60) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL9462735 0.76 HTR6 (0.68) HTR6HTR1AHTR2CDRD3HTR7
SCHEMBL12177017 0.75 KDM4E (0.64) HTR7KDM4EALDH1A1
SCHEMBL9147029 0.73 HTR6 (0.56) HTR6
SCHEMBL9149499 0.73 HTR6 (0.52) HTR6HTR1AHTR2CDRD3KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
EP-0923575-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS Takeda Chemical Industries, Ltd. (JP) 1999-06-23 EP disclosed
WO-1998008842-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-05 WO disclosed