SCHEMBL6984988

SCHEMBL6984988

CCN(Cc1ccc(F)c(Br)c1)C(=O)/C=C(\O)C(=O)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MITF O75030 1/20 0.41
HTT P42858 1/20 0.41
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MAOA P21397 3/20 0.34
MAOB P27338 3/20 0.34
BCHE P06276 2/20 0.34
ACHE P22303 2/20 0.34
TSHR P16473 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LPAR1 Q92633 1/20 0.34
LPAR5 Q9H1C0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984991 1.00 NPSR1 (0.42) NPSR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6076892 0.87 NPSR1 (0.40) NPSR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6076896 0.87 NPSR1 (0.40) NPSR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6413079 0.86 NPSR1 (0.41) NPSR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6413074 0.86 NPSR1 (0.41) NPSR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6412651 0.83 ALDH1A1 (0.46) ALDH1A1HDAC1HDAC6MAOAMAOB
SCHEMBL6412647 0.83 ALDH1A1 (0.46) ALDH1A1HDAC1HDAC6MAOAMAOB
SCHEMBL6411640 0.80 PTPN1 (0.40) KDM4EALDH1A1MITFHTTLPAR1
SCHEMBL6411635 0.80 PTPN1 (0.40) KDM4EALDH1A1MITFHTTLPAR1
SCHEMBL6879322 0.78 NPSR1 (0.41) NPSR1CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322599-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-02 EP disclosed
WO-2001096283-A9 HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2002-10-17 WO disclosed
WO-2001096283-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-12-20 WO disclosed