SCHEMBL6985071

SCHEMBL6985071

Fc1cc[c]c(C(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.36
TDO2 P48775 3/20 0.36
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
GBA1 P04062 2/20 0.32
EPHX1 P07099 1/20 0.31
NFE2L2 Q16236 1/20 0.31
CFTR P13569 1/20 0.31
GOPC Q9HD26 1/20 0.31
CNR2 P34972 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2A6 P11509 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27971479 0.80 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL3840841 0.73 DPP4 (0.40) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL1069182 0.73
SCHEMBL207047 0.71 CYP1A2 (0.30) CYP1A2CYP2A6
SCHEMBL11069143 0.70 DPP4 (0.42) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL8326680 0.68 ERAP1 (0.37) IDO1TDO2GBA1CYP2A6
SCHEMBL10406453 0.68 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL15464082 0.67 ADRA2A (0.36) IDO1TDO2SLC6A4
SCHEMBL15464250 0.67 ADRA2A (0.36) IDO1TDO2SLC6A4
SCHEMBL26232354 0.66 IDO1 (0.48) IDO1TDO2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294695-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-03-26 EP claimed
WO-2001085694-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-11-15 WO claimed
EP-1294695-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-03-26 EP disclosed
WO-2001085694-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-11-15 WO disclosed