SCHEMBL6985278

SCHEMBL6985278

COC(=O)Oc1ccc2c(c1)CCCN2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
KDM4E B2RXH2 2/20 0.52
GAA P10253 2/20 0.52
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
PPARG P37231 4/20 0.46
PPARD Q03181 4/20 0.46
PPARA Q07869 4/20 0.46
HRH3 Q9Y5N1 2/20 0.45
PLAU P00749 1/20 0.43
HSD17B10 Q99714 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP1 P29466 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384052 0.85 MAPT (0.55) MAPTKDM4EGAACA12CA1
SCHEMBL30529634 0.85 MAPT (0.55) MAPTKDM4EGAACA12CA1
Hydrochloric Acid SCHEMBL27745533 0.84 MAPT (0.54) MAPTKDM4EGAACA12CA1
SCHEMBL10909390 0.82 KDM4E (0.50) MAPTKDM4EGAACA12CA1
SCHEMBL27510896 0.82 KDM4E (0.51) MAPTKDM4EGAACA12CA1
SCHEMBL665048 0.80 CA12 (0.53) MAPTKDM4EGAACA12CA1
Hydrochloric Acid SCHEMBL8021718 0.79 KDM4E (0.53) MAPTKDM4EGAACA12CA1
SCHEMBL7336195 0.79 PPARG (0.53) MAPTKDM4EPPARGPPARDPPARA
SCHEMBL6890994 0.79 POLB (0.54) MAPTKDM4EPPARGPPARDPPARA
SCHEMBL1495030 0.78 MAPT (0.50) MAPTKDM4EGAACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed