SCHEMBL6985338

SCHEMBL6985338

O=C(OCc1ccccc1)c1cc2cc(O)ccc2o1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.66
FLT3 P36888 2/20 0.58
LMNA P02545 3/20 0.55
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
GLA P06280 1/20 0.55
GAA P10253 1/20 0.55
HPGD P15428 1/20 0.55
CASP1 P29466 1/20 0.55
BRCA1 P38398 1/20 0.55
CASP7 P55210 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
HSD17B10 Q99714 1/20 0.55
CLK1 P49759 2/20 0.52
DYRK1A Q13627 2/20 0.52
DYRK1B Q9Y463 2/20 0.52
MAPT P10636 1/20 0.52
HTT P42858 1/20 0.52
TSHR P16473 1/20 0.51
KMT2A Q03164 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717367 0.87 KMT2A (0.55) AKR1B1LMNAKDM4EALDH1A1GAA
SCHEMBL21187892 0.87 MAPT (0.68) AKR1B1FLT3KDM4EALDH1A1HPGD
SCHEMBL22479070 0.86 AKR1B1 (0.53) AKR1B1LMNAKDM4EALDH1A1CASP1
SCHEMBL22479063 0.86 PIM1 (0.60) AKR1B1LMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL6622934 0.86 MAPT (0.53) AKR1B1LMNAKDM4EALDH1A1HPGD
SCHEMBL4924372 0.86 AKR1B1 (0.53) AKR1B1KDM4EALDH1A1MAPTHTT
SCHEMBL6624774 0.84 AKR1B1 (0.51) AKR1B1LMNAKDM4EALDH1A1CASP1
SCHEMBL6981476 0.83 MAPT (0.50) AKR1B1LMNAKDM4EALDH1A1HPGD
SCHEMBL15714290 0.83 PIM1 (0.63) AKR1B1LMNAMAPTHTTTSHR
SCHEMBL1473963 0.82 MAOB (0.68) AKR1B1FLT3LMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed