SCHEMBL6985448

SCHEMBL6985448

O=[N+]([O-])c1cccc([N]c2ccccc2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.59
LMNA P02545 2/20 0.59
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
CASP3 P42574 1/20 0.56
SENP8 Q96LD8 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
SENP6 Q9GZR1 1/20 0.56
ALDH1A1 P00352 6/20 0.56
KMT2A Q03164 5/20 0.55
MEN1 O00255 3/20 0.55
NFE2L2 Q16236 1/20 0.53
HTR3E A5X5Y0 1/20 0.53
HTR3B O95264 1/20 0.53
HTR3A P46098 1/20 0.53
HTR3D Q70Z44 1/20 0.53
HTR3C Q8WXA8 1/20 0.53
MAPT P10636 1/20 0.50
MAPK1 P28482 1/20 0.50
ACHE P22303 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3189908 0.94 TSHR (0.67) TSHRLMNANPC1RAB9ACASP3
SCHEMBL1405402 0.85 NPC1 (0.65) TSHRLMNANPC1RAB9ACASP3
SCHEMBL1405403 0.85 NPC1 (0.65) TSHRLMNANPC1RAB9ACASP3
SCHEMBL7086378 0.82 ALDH1A1 (0.62) LMNANPC1RAB9ACASP3SENP8
SCHEMBL1405486 0.82 TSHR (0.67) TSHRLMNANPC1RAB9ACASP3
SCHEMBL1405487 0.82 TSHR (0.67) TSHRLMNANPC1RAB9ACASP3
SCHEMBL11359659 0.80 TSHR (0.64) TSHRLMNANPC1RAB9ACASP3
SCHEMBL7335956 0.80 TSHR (0.64) TSHRLMNANPC1RAB9ACASP3
Dinitrophenylene SCHEMBL27707690 0.79 TSHR (0.85) TSHRLMNANPC1RAB9AALDH1A1
Dinitrophenylene SCHEMBL27564057 0.79 TSHR (0.94) TSHRLMNAALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294695-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-03-26 EP claimed
WO-2001085694-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-11-15 WO claimed
EP-1294695-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-03-26 EP disclosed
WO-2001085694-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-11-15 WO disclosed