SCHEMBL6985863

SCHEMBL6985863

Nc1nc(N)nc(C2(c3ccccc3)CCCCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALOX5AP P20292 2/20 0.42
HSD11B1 P28845 2/20 0.40
HSD11B2 P80365 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DPP4 P27487 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
HSD17B10 Q99714 1/20 0.38
POLB P06746 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116796 0.87 ALDH1A1 (0.40) ALDH1A1L3MBTL1ALOX5APMEN1KMT2A
SCHEMBL6980554 0.79 BACE1 (0.58) ALDH1A1L3MBTL1
SCHEMBL30078304 0.76 ESR1 (0.58) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL54982 0.76 ESR1 (0.58) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL28378542 0.76 ESR1 (0.58) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL24157288 0.76 ESR1 (0.58) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL30877902 0.76 ESR1 (0.58) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL30877914 0.76 ESR1 (0.58) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL9607808 0.75 CSNK1A1 (0.42) ALDH1A1L3MBTL1HSD11B1HSD11B2MEN1
Ammonia Solution, Strong SCHEMBL7989528 0.74 ESR1 (0.56) ALDH1A1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037886-B1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LAB (US) 2003-05-02 EP claimed
US-6288228-B1 DIAMINOTRIAZINE DERIVATIVES ABBOTT LABORATORIES 2001-09-11 US claimed
US-6150362-A ADMINISTERING 1,3,5-SUBSTITUTED TRIAZINE COMPOUNDS TO THE PATIENT SUFFERING FROM ANGIOGENIC DISEASES ABBVIE INC. 2000-11-21 US claimed
EP-1037886-A1 TRIAZINE ANGIOGENESIS INHIBITORS Abbott Laboratories (US) 2000-09-27 EP claimed
WO-1999031088-A1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LABORATORIES (US) 1999-06-24 WO claimed
EP-1037886-B1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LAB (US) 2003-05-02 EP disclosed
US-6288228-B1 DIAMINOTRIAZINE DERIVATIVES ABBOTT LABORATORIES 2001-09-11 US disclosed
US-6150362-A ADMINISTERING 1,3,5-SUBSTITUTED TRIAZINE COMPOUNDS TO THE PATIENT SUFFERING FROM ANGIOGENIC DISEASES ABBVIE INC. 2000-11-21 US disclosed
EP-1037886-A1 TRIAZINE ANGIOGENESIS INHIBITORS Abbott Laboratories (US) 2000-09-27 EP disclosed
WO-1999031088-A1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LABORATORIES (US) 1999-06-24 WO disclosed