SCHEMBL6987162

SCHEMBL6987162

COc1ccc(C(=O)c2ccsc2NCC(=O)NCC2CCNCC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 2/20 0.44
HTR4 Q13639 2/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM1A O60341 1/20 0.39
MAPK8 P45983 1/20 0.39
KDM4E B2RXH2 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
LMNA P02545 1/20 0.37
CHRM1 P11229 1/20 0.37
FAAH O00519 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982744 0.85 EP300 (0.45) EP300HTR4NPC1RAB9AALDH1A1
Hydrochloric Acid SCHEMBL6982028 0.84 NPC1 (0.40) HTR4NPC1RAB9AALDH1A1MAPK8
SCHEMBL6990414 0.80 HTR4 (0.43) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6985733 0.80 HTR4 (0.43) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6989025 0.80 HTR4 (0.43) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6985413 0.79 HTR4 (0.43) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6986612 0.79 HTR4 (0.43) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6983529 0.78 HTR4 (0.42) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6987917 0.78 HTR4 (0.42) EP300HTR4NPC1ALDH1A1SMN1; SMN2
SCHEMBL6990268 0.77 HTR4 (0.41) EP300HTR4NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289954-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096303-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed