SCHEMBL6987263

SCHEMBL6987263

CNC(=O)N1N=C(c2ccc([N+](=O)[O-])cc2)c2cc3c(cc2C[C@H]1C)OCO3

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.76
GRIA2 P42262 1/20 0.76
BRD4 O60885 5/20 0.50
TERT O14746 3/20 0.49
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B10 Q99714 2/20 0.43
THRB P10828 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8793610 1.00 GRIA1 (0.76) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL6615773 0.90 GRIA1 (0.60) GRIA1GRIA2TERTMEN1KMT2A
SCHEMBL6991386 0.90 GRIA1 (0.60) GRIA1GRIA2TERTMEN1KMT2A
SCHEMBL5429840 0.90 GRIA1 (0.60) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL5881337 0.89 GRIA1 (0.71) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL7226682 0.88 GRIA1 (0.60) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL5416041 0.88 GRIA1 (0.59) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL5416047 0.88 GRIA1 (0.59) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL5433568 0.87 GRIA1 (0.58) GRIA1GRIA2BRD4TERTMEN1
SCHEMBL8793131 0.87 GRIA1 (0.59) GRIA1GRIA2BRD4TERTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0699677-B1 Stereoselective process for producing dihydro-2,3-benzodiazepine derivatives LILLY CO ELI (US) 2003-01-29 EP disclosed
US-6160133-A Synthesis of (S)-α-methyl-1,3-benzodioxole-5-ethanol and derivatives ELI LILLY AND COMPANY (US) 2000-12-12 US disclosed
US-5986114-A MUSCLE RELAXANTS, NERVOUS SYSTEM DISORDERS OR ANTICONVULSANTS ELI LILLY AND COMPANY (US) 1999-11-16 US disclosed
US-5665878-A Stereoselective process for producing dihydro-2,3-benzodiazepine derivatives ELI LILLY AND COMPANY (US) 1997-09-09 US disclosed
EP-0699677-A1 Stereoselective process for producing dihydro-2,3-benzodiazepine derivatives ELI LILLY AND COMPANY (US) 1996-03-06 EP disclosed