SCHEMBL6988742

SCHEMBL6988742

O=CCN1CC(c2ccccc2)CC1=O

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.67
HPGD P15428 1/20 0.67
TP53 P04637 1/20 0.56
CHRM2 P08172 1/20 0.56
CHRM4 P08173 1/20 0.56
CHRM5 P08912 1/20 0.56
CHRM1 P11229 1/20 0.56
CHRM3 P20309 1/20 0.56
BRD4 O60885 4/20 0.56
ALDH1A1 P00352 2/20 0.49
PKM P14618 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 1/20 0.46
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13533665 1.00 TSHR (0.67) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL13533666 1.00 TSHR (0.67) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL10760741 0.87 TSHR (0.63) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL10762307 0.81 HPGD (0.69) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL13532862 0.81 HPGD (0.69) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL2958047 0.81 TSHR (0.69) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL11471890 0.81 HPGD (0.73) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL11472575 0.81 TSHR (0.69) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL16033027 0.80 HPGD (1.00) TSHRHPGDTP53CHRM2CHRM4
SCHEMBL10755797 0.79 HPGD (0.65) TSHRHPGDTP53CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061472-A A pharmaceutical composition in the form of tablet and its preparation method “瓦连塔印铁列克特”有限公司 2016-10-26 CN claimed
EP-1326829-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE-II INHIBITORS Bayer Pharmaceuticals Corporation (US) 2003-07-16 EP disclosed
WO-2002026706-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE-II INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2002-04-04 WO disclosed