SCHEMBL6988951

SCHEMBL6988951

CC(=O)ON(C)C(=O)C#Cc1ccccc1F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.38
GRM5 P41594 5/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
MME P08473 3/20 0.34
ECE1 P42892 3/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
IKBKB O14920 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
VCP P55072 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28722215 0.76 GRM5 (0.44) GRM5PTGDR2MMEECE1HCAR2
SCHEMBL6768178 0.71 CA12 (0.40) NPSR1GRM5MEN1KMT2AKDM4E
SCHEMBL15841080 0.71 GRM5 (0.41) GRM5PTGDR2MMEECE1MEN1
SCHEMBL4174272 0.70 MLYCD (0.44) NPSR1MMEECE1KMT2AKDM4E
SCHEMBL6773718 0.70 PTGDR2 (0.43) GRM5PTGDR2MMEECE1HCAR2
SCHEMBL30467436 0.70 PTGDR2 (0.43) GRM5PTGDR2MMEECE1HCAR2
SCHEMBL31182405 0.69 GRM5 (0.44) GRM5PTGDR2MMEECE1IKBKB
SCHEMBL15062326 0.68 NPSR1 (0.68) NPSR1MEN1KMT2AKDM4ENPC1
SCHEMBL6774626 0.68 GRM5 (0.46) GRM5PTGDR2MMEECE1MEN1
SCHEMBL28499185 0.66 GRM5 (0.38) GRM5PTGDR2MMEECE1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326829-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE-II INHIBITORS Bayer Pharmaceuticals Corporation (US) 2003-07-16 EP disclosed
WO-2002026706-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE-II INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2002-04-04 WO disclosed