Bicarbonate

Bicarbonate

SCHEMBL6989679

COc1cc(C)c(CC(=O)NC2CCC(C)CC2)c(C)c1.O=C(O)O

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
EPHX2 P34913 1/20 0.45
SIGMAR1 Q99720 2/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL6995801 0.89 EPHX2 (0.57) LMNASMN1; SMN2EPHX2SIGMAR1MEN1
Bicarbonate SCHEMBL7000560 0.88 EPHX2 (0.44) SMN1; SMN2EPHX2SIGMAR1CNR1CNR2
Bicarbonate SCHEMBL6998472 0.88 EPHX2 (0.59) LMNASMN1; SMN2EPHX2MEN1KMT2A
Bicarbonate SCHEMBL7000575 0.88 EPHX2 (0.59) LMNASMN1; SMN2EPHX2MEN1KMT2A
Bicarbonate SCHEMBL6991031 0.87 KMT2A (0.50) SMN1; SMN2EPHX2SIGMAR1CNR1CNR2
Bicarbonate SCHEMBL7615552 0.86 EPHX2 (0.46) GAALMNAMAPK1SMN1; SMN2EPHX2
Bicarbonate SCHEMBL6996297 0.86 SIGMAR1 (0.40) GAASMN1; SMN2EPHX2SIGMAR1CNR1
Bicarbonate SCHEMBL6996202 0.86 SIGMAR1 (0.42) SMN1; SMN2EPHX2SIGMAR1CNR1CNR2
Bicarbonate SCHEMBL6991552 0.86 MEN1 (0.44) GAAEPHX2SIGMAR1CNR1CNR2
Bicarbonate SCHEMBL6989581 0.85 EPHX2 (0.44) SMN1; SMN2EPHX2SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0754175-B1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER CROPSCIENCE AG (DE) 2003-01-29 EP disclosed
EP-0754175-A1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER AG (DE) 1997-01-22 EP disclosed
WO-1995026954-A1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1995-10-12 WO disclosed