SCHEMBL6989870

SCHEMBL6989870

COc1ccc2c(Nc3ccc4c(c3)NCC4)c(C#N)cnc2c1OC

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.49
ERBB2 P04626 10/20 0.49
SRC P12931 7/20 0.49
GAK O14976 1/20 0.45
MAP2K1 Q02750 3/20 0.44
PRKCQ Q04759 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999979 0.87 EGFR (0.44) EGFRERBB2SRCMAP2K1
SCHEMBL6997455 0.87 MAP2K1 (0.42) EGFRERBB2SRCMAP2K1PRKCQ
SCHEMBL4455183 0.84 EGFR (0.69) EGFRERBB2SRCMAP2K1
SCHEMBL6381073 0.83 EGFR (0.69) EGFRERBB2SRCGAKMAP2K1
SCHEMBL6998602 0.81 MAP2K1 (0.62) EGFRERBB2SRCMAP2K1
SCHEMBL6382800 0.80 EGFR (0.56) EGFRERBB2SRCGAKMAP2K1
SCHEMBL6379771 0.80 SRC (0.61) EGFRERBB2SRCGAKMAP2K1
SCHEMBL6385365 0.79 EGFR (0.69) EGFRERBB2SRCGAKMAP2K1
SCHEMBL6379913 0.79 EGFR (0.65) EGFRERBB2SRCGAKMAP2K1
SCHEMBL7003514 0.78 PRKCQ (0.59) EGFRERBB2SRCGAKMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117659-B1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS WYETH CORP (US) 2003-12-03 EP claimed